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Found 2 Enz. Inhib. hit(s) with Target = 'Neuromedin-U receptor 1' and Ligand = 'BDBM50291671'
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50291671(CHEMBL4166325)
Affinity DataIC50:  54nMAssay Description:Compound was tested for in vitro motilin receptor binding affinityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50291671(CHEMBL4166325)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed