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Found 2 Enz. Inhib. hit(s) with Target = 'Neutrophil elastase' and Ligand = 'BDBM50036049'
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50036049(((S)-1-{(S)-2-[(S)-1-(4,5-Dihydro-oxazole-2-carbon...)
Affinity DataKi:  0.550nMAssay Description:In vitro inhibitory activity against human neutrophil elastase (HNE) catalyzed hydrolysis of the synthetic substrate MeO-Suc-Ala- Ala-Pro-Val-pNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50036049(((S)-1-{(S)-2-[(S)-1-(4,5-Dihydro-oxazole-2-carbon...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed