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Found 2 Enz. Inhib. hit(s) with Target = 'Nicotinamide phosphoribosyltransferase' and Ligand = 'BDBM50117198'
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Kyowa Hakko Kogyo

LigandPNGBDBM50117198(4-{[7-Chloro-3-methyl-2-(4-methyl-piperazin-1-ylme...)
Affinity DataIC50:  0.230nMAssay Description:In vitro inhibition assay using human nampt, NMN adenylytransferase (nmant1)and UDP-glucose dehdryogenase (ugdh) genes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Kyowa Hakko Kogyo

LigandPNGBDBM50117198(4-{[7-Chloro-3-methyl-2-(4-methyl-piperazin-1-ylme...)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of nicotinamide phosphoribosyltransferase-catalyzed conversion of nicotinamide to nicotinamide mononucleotideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed