Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Nociceptin receptor' and Ligand = 'BDBM50274460'
TargetNociceptin receptor(Mouse)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50274460(CHEMBL504540 | FGGFTGARKSARKYANQ | OFQ/N,[Tyr14])
Affinity DataKi:  0.00700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNociceptin receptor(Mouse)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50274460(CHEMBL504540 | FGGFTGARKSARKYANQ | OFQ/N,[Tyr14])
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNociceptin receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50274460(CHEMBL504540 | FGGFTGARKSARKYANQ | OFQ/N,[Tyr14])
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50274460(CHEMBL504540 | FGGFTGARKSARKYANQ | OFQ/N,[Tyr14])
Affinity DataEC50:  11nMAssay Description:Activation of rat ORL1 receptor expressed in african green monkey COS7 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed