Found 1 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50233305'
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)
Curated by ChEMBL
Wuxi Apptec (Shanghai)
Curated by ChEMBL
Affinity DataIC50: 5.02E+3nMAssay Description:Antagonist activity at human orexin 1 receptor expressed in HEK293 cells assessed as inhibition of orexin-induced calcium mobilization after 60 mins ...More data for this Ligand-Target Pair