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Found 2 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50454547'
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454547(CHEMBL4213974)
Affinity DataKi:  2.10nMAssay Description:Antagonist activity at human OX1R expressed in CHOK1 cells assessed as inhibition of orexin A-induced intracellular Ca2+ release preincubated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454547(CHEMBL4213974)
Affinity DataKi:  2.30nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed