Found 2 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50592808'
Affinity DataKi: 11.7nMAssay Description:Antagonist activity at human OX1R expressed in CHO-K1 cells assessed as inhibition of orexin-A-induced increase in calcium mobilization preincubated ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at human OX1R expressed in CHO-K1 cells assessed as inhibition of orexin-A-induced increase in calcium mobilization preincubated ...More data for this Ligand-Target Pair