Affinity DataKi: 500nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair