Affinity DataKi: 86nMAssay Description:Displacement of [33P]2-MeS-ADP from human recombinant P2Y12 receptor expressed in CHO cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human P2Y12More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of ADP-induced platelet aggregation measured for 5 mins by lig...More data for this Ligand-Target Pair
![](/img/powered_by_small.gif)