Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM21785'
LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  3.45E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  2.90E+3nMT: 2°CAssay Description:Activity was assessed by measuring the human PPAR ligand binding domain with the co-activator protein. Europium labeled anti-GST antibody, streptavid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed