Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50121416'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 6.70E+4nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair