Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50135777'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135777(2-(4-{3-[1-(4-tert-Butyl-benzyl)-4-methyl-5-oxo-4,...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135777(2-(4-{3-[1-(4-tert-Butyl-benzyl)-4-methyl-5-oxo-4,...)
Affinity DataIC50:  15nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135777(2-(4-{3-[1-(4-tert-Butyl-benzyl)-4-methyl-5-oxo-4,...)
Affinity DataEC50:  2nMAssay Description:Cotransfection activity against human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed