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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50200402'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50: >6.00E+3nMAssay Description:Activity at human PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed