Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50519891'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519891(CHEMBL4452679)
Affinity DataIC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed