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Found 2 Enz. Inhib. hit(s) with Target = 'Probable G-protein coupled receptor 142' and Ligand = 'BDBM332764'
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Lilly China Research and Development Center (Lcrdc)

Curated by ChEMBL
LigandPNGBDBM332764(Cis-(chiral)-3-Chloro-N-[2- [5-(1,4-dimethyl-1H- i...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Lilly China Research and Development Center (Lcrdc)

Curated by ChEMBL
LigandPNGBDBM332764(Cis-(chiral)-3-Chloro-N-[2- [5-(1,4-dimethyl-1H- i...)
Affinity DataEC50:  27.2nMAssay Description:HEK293 cells expressing human GPR142 are maintained in DMEM supplemented with 10% FBS and 800 μg/ml G418 (Geneticin) at 37° C. and 5% CO2. The c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent