TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity against CRTh2 receptor in human eosinophils assessed as cell shape changeMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 311nMAssay Description:Antagonist activity against human CRTh2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair