Report error Found 2 Enz. Inhib. hit(s) with Target = 'Prostaglandin D2 receptor 2' and Ligand = 'BDBM50387201'
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human CRTh2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human CRTh2 receptor expressed in HEK293 cells assessed as inhibition of PGD2-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair