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Found 3 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP2 subtype' and Ligand = 'BDBM85602'
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by PDSP Ki Database
LigandPNGBDBM85602((R)-BUTAPROST | Butaprost (Free Acid) | CAS_69648-...)
Affinity DataKi:  91nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by PDSP Ki Database
LigandPNGBDBM85602((R)-BUTAPROST | Butaprost (Free Acid) | CAS_69648-...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to EP2 receptor (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by PDSP Ki Database
LigandPNGBDBM85602((R)-BUTAPROST | Butaprost (Free Acid) | CAS_69648-...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at EP2 receptor (unknown origin) by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed