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Report error Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50520989'
LigandPNGBDBM50520989(CHEMBL4565280)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of human recombinant FTase using [3H]FPP as substrate after 15 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed