Report error Found 20 Enz. Inhib. hit(s) with Target = 'Proto-oncogene tyrosine-protein kinase Src' and Ligand = 'BDBM2579'
Affinity DataIC50: 0.830nMAssay Description:Inhibition of c-Src using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of src kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of c-SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human c-SRC using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of SRC (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human c-SRC using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of c-Src (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of SRC (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human Src expressed in insect cells using Ulight-Poly GAT[EAY(1:1:1)]n as substrate after 10 mins by LANCE methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Chicken)
Chemical Genomics Centre of The Max Planck Society
Chemical Genomics Centre of The Max Planck Society
Affinity DataIC50: 6.30nM Kd: 8nMAssay Description:Tyrosine kinase inhibition assay using wild type cSrc measured by a fluorescence-labeled approach.More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of recombinant human Src using Ulight-Poly GAT[EAY(1:1:1)]n as substrate measured after 10 mins by LANCE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human Src kinase by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
Affinity DataKd: 86nMAssay Description:Binding constant for SRC kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Average Binding Constant for SRC; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 86nMAssay Description:Binding constant for SRC kinase domainMore data for this Ligand-Target Pair