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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'RAC-beta serine/threonine-protein kinase' and Ligand = 'BDBM16219'
Target
RAC-beta serine/threonine-protein kinase
(Homo sapiens (Human))
Astex
Ligand
BDBM16219
(4-(4-chlorophenyl)-4-[4-(1H-pyrazol-4-yl)phenyl]pi...)
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Affinity Data
IC50: 18nM
pH: 7.2 T: 2°C
Assay Description:
The purified PKB beta enzyme was assayed with a peptide substrate and test compound in the presence of 30 uM ATP/ [gamma-33P]ATP in 96-well plates. I...
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