Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1' and Ligand = 'BDBM50195202'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195202(3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(2H-1...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human CHEK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195202(3-(5-(piperidin-1-ylmethyl)-1H-indol-2-yl)-6-(2H-1...)
Affinity DataEC50:  880nMAssay Description:Release of camptothecin-induced cell cycle arrest in NCI-H1299 cells mediated by CHEK1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed