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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK1' and Ligand = 'BDBM28171'
Target
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human))
Gsk
Ligand
BDBM28171
(3-[(2-bromophenyl)methoxy]-5-[6-(trifluoromethyl)-...)
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Affinity Data
IC50: 9nM
pH: 7.2 T: 2°C
Assay Description:
The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...
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