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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK1' and Ligand = 'BDBM50263741'
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Rockefeller University

Curated by ChEMBL
LigandPNGBDBM50263741(5-Cyano-7-nitro-3-oxy-benzothiazole-2-carboxylic a...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of recombinant polo-like kinase 1 activity by SDS-PAGEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Rockefeller University

Curated by ChEMBL
LigandPNGBDBM50263741(5-Cyano-7-nitro-3-oxy-benzothiazole-2-carboxylic a...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed