Found 6 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 8 subunit alpha' and Ligand = 'BDBM50558815'
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells incubated for 30 mins by FLIPRTetra fluorescent membrane potential assayMore data for this Ligand-Target Pair
Ligand InfoKEGG
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 72.4nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells incubated for 30 mins by FLIPRTetra fluorescent membrane potential assayMore data for this Ligand-Target Pair
Ligand InfoKEGG
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 6.30nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells assessed as decrease in peak current at pulses to 0 mV by whole cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoKEGG
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 72.4nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells incubated for 30 mins by FLIPRTetra fluorescent membrane potential assayMore data for this Ligand-Target Pair
Ligand InfoKEGG
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 6.20nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells assessed as decrease in peak current at pulses to 0 mV by whole cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoKEGG
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells incubated for 30 mins by FLIPRTetra fluorescent membrane potential assayMore data for this Ligand-Target Pair
Ligand InfoKEGG