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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50099304'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099304(CHEMBL275541 | [(3S,4R)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]DA uptake at Dopamine transporter in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099304(CHEMBL275541 | [(3S,4R)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataIC50:  46nMAssay Description:Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptake at a concentration of 30 nM with cocaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099304(CHEMBL275541 | [(3S,4R)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataIC50:  308nMAssay Description:Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099304(CHEMBL275541 | [(3S,4R)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataIC50:  641nMAssay Description:Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptake at a concentration of 100 nM with cocaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed