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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent noradrenaline transporter' and Ligand = 'BDBM50400815'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50400815((S)-VENLAFAXINE | VENLAFAXINE)
Affinity DataIC50:  149nMAssay Description:Inhibition of NET (unknown origin) assessed as noradrenaline reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50400815((S)-VENLAFAXINE | VENLAFAXINE)
Affinity DataIC50:  754nMAssay Description:Inhibition of human NET expressed in MDCK cells assessed as decrease in [3H]-noradrenaline reuptake after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50400815((S)-VENLAFAXINE | VENLAFAXINE)
Affinity DataIC50:  754nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed