Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent noradrenaline transporter' and Ligand = 'BDBM50400815'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis
Curated by ChEMBL
University Of California Davis
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Inhibition of NET (unknown origin) assessed as noradrenaline reuptakeMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis
Curated by ChEMBL
University Of California Davis
Curated by ChEMBL
Affinity DataIC50: 754nMAssay Description:Inhibition of human NET expressed in MDCK cells assessed as decrease in [3H]-noradrenaline reuptake after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of California Davis
Curated by ChEMBL
University Of California Davis
Curated by ChEMBL