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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK [357-620,Y512E]' and Ligand = 'BDBM213221'
Target
Tyrosine-protein kinase ITK/TSK [357-620,Y512E]
(Homo sapiens (Human))
Glaxosmithkline
Ligand
BDBM213221
((S)-1-(3-((4-(Piperidin-1-ylmethyl)-6-(thiazolo[5,...)
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Affinity Data
IC50: 6.30nM
Assay Description:
This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...
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Target Info
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Ligand Info
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