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Found 4 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50262270'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  388nMAssay Description:Antagonist activity at vassopressin V1a receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  388nMAssay Description:Displacement of [3H]-vasopressin from human vasopressin V1a receptor expressed in CHO cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  388nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  388nMAssay Description:Antagonist activity at human cloned vasopressin V1A receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed