Report error Found 9 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM50205990'
Affinity DataKi: 61nMAssay Description:Binding affinity against Vasopressin receptor in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Binding affinity against Vasopressin receptor in rat kidney medullaMore data for this Ligand-Target Pair
Affinity DataKi: 1.54E+3nMAssay Description:Binding affinity to V2R (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity towards human Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at human kidney vasopressin V2 receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 min...More data for this Ligand-Target Pair
Affinity DataEC50: 810nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair