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Report error Found 2 Enz. Inhib. hit(s) with Target = 'cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A' and Ligand = 'BDBM50398011'
LigandPNGBDBM50398011(CHEMBL2180423 | US8492392, O-2)
Affinity DataKi:  0.920nMAssay Description:Inhibition of PDE10A by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50398011(CHEMBL2180423 | US8492392, O-2)
Affinity DataKi:  0.930nM ΔG°:  -51.5kJ/moleT: 25°CAssay Description:Fluorescence polarization assay: The compounds of the following examples had activity in reference assays by exhibiting the ability to inhibit the hy...More data for this Ligand-Target Pair
In DepthDetails US Patent