BindingDB PrimarySearch_ki

Found 52 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50009645

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 22nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 22nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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PDB

3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 27nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 27nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 48nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 48nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530632(CHEMBL4458437)

IC50: 117nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530632(CHEMBL4458437)

IC50: 117nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530624(CHEMBL4463012)

IC50: 131nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530624(CHEMBL4463012)

IC50: 131nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530630(CHEMBL2310642)

IC50: 147nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530630(CHEMBL2310642)

IC50: 147nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 157nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 157nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530631(CHEMBL4583178)

IC50: 283nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530631(CHEMBL4583178)

IC50: 283nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 500nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 500nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 650nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 650nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530619(CHEMBL4446953)

IC50: 779nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530619(CHEMBL4446953)

IC50: 779nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530616(CHEMBL4450843)

IC50: 1.06E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530616(CHEMBL4450843)

IC50: 1.06E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530628(CHEMBL4475546)

IC50: 1.08E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530628(CHEMBL4475546)

IC50: 1.08E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530634(CHEMBL4447962)

IC50: 1.26E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530634(CHEMBL4447962)

IC50: 1.26E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530635(CHEMBL4448691)

IC50: 1.32E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530635(CHEMBL4448691)

IC50: 1.32E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530629(CHEMBL4556670)

IC50: 2.32E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530629(CHEMBL4556670)

IC50: 2.32E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530626(CHEMBL4447036)

IC50: 2.46E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530626(CHEMBL4447036)

IC50: 2.46E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530620(CHEMBL4447289)

IC50: 4.63E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530620(CHEMBL4447289)

IC50: 4.63E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530627(CHEMBL4456359)

IC50: 6.37E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530627(CHEMBL4456359)

IC50: 6.37E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)

IC50: 6.75E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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MMDB
PDB

3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)

IC50: 6.75E+3nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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MMDB
PDB

3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530636(CHEMBL4441440)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530625(CHEMBL4527132)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322820(CHEMBL1172781 | S-2-(5,6-Diphenylfuro[2,3-d]pyrimi...)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530617(CHEMBL4448148)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530636(CHEMBL4441440)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530621(CHEMBL4565374)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530625(CHEMBL4527132)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530621(CHEMBL4565374)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530633(CHEMBL4531827)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530617(CHEMBL4448148)

IC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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