Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50016866
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597908(CHEMBL5181496)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597908(CHEMBL5181496)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597906(CHEMBL5183539)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597916(CHEMBL5201115)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597916(CHEMBL5201115)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597896(CHEMBL5181996)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597896(CHEMBL5181996)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597913(CHEMBL5194549)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597913(CHEMBL5194549)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597915(CHEMBL5185237)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597915(CHEMBL5185237)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597909(CHEMBL5196929)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597909(CHEMBL5196929)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597904(CHEMBL5176448)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597905(CHEMBL5182266)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597905(CHEMBL5182266)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597904(CHEMBL5176448)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597907(CHEMBL5189879)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597914(CHEMBL5188480)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597914(CHEMBL5188480)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597902(CHEMBL5177632)
Affinity DataIC50:  4nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597912(CHEMBL5196259)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597912(CHEMBL5196259)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597910(CHEMBL5202219)
Affinity DataIC50:  10nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597910(CHEMBL5202219)
Affinity DataIC50:  10nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597898(CHEMBL5172378)
Affinity DataIC50:  13nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597911(CHEMBL5171701)
Affinity DataIC50:  13nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597911(CHEMBL5171701)
Affinity DataIC50:  13nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597898(CHEMBL5172378)
Affinity DataIC50:  13nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597895(CHEMBL5189798)
Affinity DataIC50:  26nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597895(CHEMBL5189798)
Affinity DataIC50:  26nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597903(CHEMBL5197729)
Affinity DataIC50:  36nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597900(CHEMBL5194727)
Affinity DataIC50:  43nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597901(CHEMBL5192632)
Affinity DataIC50:  66nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597890(CHEMBL5205566)
Affinity DataIC50:  90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597890(CHEMBL5205566)
Affinity DataIC50:  90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597894(CHEMBL5187919)
Affinity DataIC50:  90nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597891(CHEMBL5195100)
Affinity DataIC50:  120nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597891(CHEMBL5195100)
Affinity DataIC50:  120nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597899(CHEMBL5178518)
Affinity DataIC50:  130nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597893(CHEMBL5201671)
Affinity DataIC50:  130nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597893(CHEMBL5201671)
Affinity DataIC50:  130nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597899(CHEMBL5178518)
Affinity DataIC50:  130nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597892(CHEMBL5176666)
Affinity DataIC50:  180nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597892(CHEMBL5176666)
Affinity DataIC50:  180nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597897(CHEMBL5170393)
Affinity DataIC50:  220nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597897(CHEMBL5170393)
Affinity DataIC50:  220nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597888(CHEMBL5191174)
Affinity DataIC50:  920nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597888(CHEMBL5191174)
Affinity DataIC50:  920nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50597887(CHEMBL5196641)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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