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Found 2 Enz. Inhib. hit(s) with all data for assayid = 16 entry = 50015578
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50514200(CHEMBL4446378 | US10703733, Comparative Example 1)
Affinity DataKi:  950nMAssay Description:Inhibition of recombinant His10-tagged human Bcl-2 (2 to 211 residues) using biotinylated Bim BH3 peptide as substrate incubated for 60 mins by TR-FR...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM470606(US10821115, Example 10 | US11224601, Example 10)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of recombinant His10-tagged human Bcl-2 (2 to 211 residues) using biotinylated Bim BH3 peptide as substrate incubated for 60 mins by TR-FR...More data for this Ligand-Target Pair
In DepthDetails PubMed