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Found 27 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50045117
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045569(CHEMBL3314284)
Affinity DataIC50:  61nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045566(CHEMBL3313935)
Affinity DataIC50:  274nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045562(CHEMBL3314278)
Affinity DataIC50:  352nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045561(CHEMBL3314277)
Affinity DataIC50:  500nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045565(CHEMBL3314281)
Affinity DataIC50:  911nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045567(CHEMBL3314282)
Affinity DataIC50:  3.71E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045563(CHEMBL3314279)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045568(CHEMBL3314283)
Affinity DataIC50:  6.62E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045560(CHEMBL3314276)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045564(CHEMBL3314280)
Affinity DataIC50:  4.55E+4nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045555(CHEMBL3314271)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045556(CHEMBL3314272)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045557(CHEMBL3314273)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045558(CHEMBL3314274)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045559(CHEMBL3314275)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045570(CHEMBL3314285)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045580(CHEMBL3120970)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045579(CHEMBL3120985)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045578(CHEMBL3120969)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045577(CHEMBL3120986)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045576(CHEMBL3314270)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045575(CHEMBL3120963)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045574(CHEMBL3120983)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045573(CHEMBL3120995)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045571(CHEMBL3314286)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50044784(CHEBI:79090 | SB-202190 | US10865384, Compound SB2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Syncom

Curated by ChEMBL
LigandPNGBDBM50045572(CHEMBL3120960)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed