Report error Found 1029 with Last Name = 'inglese' and Initial = 'j'
Affinity DataKi: 14nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 21nM ΔG°: -43.2kJ/mole IC50: 31nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 52nM ΔG°: -41.0kJ/mole IC50: 103nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 55nM ΔG°: -40.9kJ/mole IC50: 133nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 56nM ΔG°: -40.8kJ/mole IC50: 63nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Pennsylvania State University
Curated by ChEMBL
Pennsylvania State University
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Compound was tested for inhibition constant against GAR TFase in miceMore data for this Ligand-Target Pair
Affinity DataKi: 102nM ΔG°: -39.4kJ/mole IC50: 168nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 120nM ΔG°: -39.0kJ/mole IC50: 268nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 121nM ΔG°: -39.0kJ/mole IC50: 183nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Competitive inhibition of recombinant Trypanosoma cruzi cruzain by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 184nM ΔG°: -37.9kJ/mole IC50: 452nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 320nM ΔG°: -36.6kJ/mole IC50: 430nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 514nM ΔG°: -35.4kJ/mole IC50: 1.06E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 556nM ΔG°: -35.2kJ/mole IC50: 1.29E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 975nM ΔG°: -33.8kJ/mole IC50: 2.45E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+3nM ΔG°: -31.3kJ/mole IC50: 4.31E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 4.23E+3nM ΔG°: -30.3kJ/mole IC50: 7.73E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 7.15E+3nM ΔG°: -29.0kJ/mole IC50: 2.46E+4nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 8.44E+3nM ΔG°: -28.6kJ/mole IC50: 2.96E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 1.34E+4nM ΔG°: -27.4kJ/mole IC50: 6.46E+3nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 1.92E+4nM ΔG°: -26.6kJ/mole IC50: 2.52E+4nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 2.34E+4nM ΔG°: -26.1kJ/mole IC50: 3.44E+4nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair
Affinity DataKi: 5.06E+4nM ΔG°: -24.2kJ/mole IC50: >1.00E+5nMpH: 5.9 T: 21°CAssay Description:Enzyme activity was determined as the production of fluorescent resorufin from the substrate. The fluorescence was measured (excitation 570 nm, emiss...More data for this Ligand-Target Pair