Compile Data Set for Download or QSAR
maximum 50k data
Found 118 of ic50 for UniProtKB: P12390
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140093(CHEMBL406720 | GCCSHPACAANNQDYC*)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140086(CHEMBL415207 | GGGCCSHPACAANNQDYC*)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587085(CHEMBL5092179)
Affinity DataIC50:  0.280nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in xenopus oocytes assessed as inhibition of Ach- induced response at -70 mV holding potential...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516324(CHEMBL4457372)
Affinity DataIC50:  0.280nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140092(CHEMBL437662 | GGCCSHPACAANNQDYC*)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516321(CHEMBL4577209)
Affinity DataIC50:  0.290nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140092(CHEMBL437662 | GGCCSHPACAANNQDYC*)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516308(CHEMBL4469829)
Affinity DataIC50:  0.380nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140087(CHEMBL265198 | GCCSNPVCHLEHSNLC*)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140088(CHEMBL451251 | GGCCSHPACAANNQDYC#)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516329(CHEMBL4467363)
Affinity DataIC50:  0.570nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140089(CHEMBL437423 | GCCSHPACAGNNQHIC*)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516323(CHEMBL4474129)
Affinity DataIC50:  1.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50547502(CHEMBL4793300)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of rat alpha3beta2 expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current response at -70 mV ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516316(CHEMBL4454928)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516325(CHEMBL4463089)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516307(CHEMBL4445542)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516337(CHEMBL4594136)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516322(CHEMBL4447464)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50554885(CHEMBL4797154)
Affinity DataIC50:  2.10nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM86240(Alpha-Conotoxin MII | Gly-L-Cys(1)-L-Cys(2)-L-Ser-...)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516343(CHEMBL4535637)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50554891(CHEMBL4753165)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516306(CHEMBL4438403)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50554892(CHEMBL4751264)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587092(CHEMBL5087554)
Affinity DataIC50:  5.70nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in xenopus oocytes assessed as inhibition of Ach- induced response at -70 mV holding potential...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140094(CCSHPACAANNQDYC* | CHEMBL262475)
Affinity DataIC50:  5.84nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587087(CHEMBL5070268)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in xenopus oocytes assessed as inhibition of Ach- induced response at -70 mV holding potential...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516342(CHEMBL4461998)
Affinity DataIC50:  6.40nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516314(CHEMBL4462168)
Affinity DataIC50:  7.10nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50554893(CHEMBL4752161)
Affinity DataIC50:  7.5nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516319(CHEMBL4443205)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516309(CHEMBL4594009)
Affinity DataIC50:  8.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516315(CHEMBL4515208)
Affinity DataIC50:  9.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516340(CHEMBL4439678)
Affinity DataIC50:  9.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516331(CHEMBL4583045)
Affinity DataIC50:  9.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140085(CHEMBL266702 | GCCSLPPCAANNPDYC*)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)
Affinity DataIC50:  9.70nMAssay Description:Inhibition of rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response by two-elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516320(CHEMBL4572578)
Affinity DataIC50:  9.80nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50140091(CHEMBL413505 | IRDgammaCCSNPACRVNNOHVC#)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in Xenopus OocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50547501(CHEMBL4788244)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat alpha3beta2 expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current response at -70 mV ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516336(CHEMBL4465982)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516313(CHEMBL4459917)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516336(CHEMBL4465982)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in xenopus oocytes assessed as inhibition of Ach- induced response at -70 mV holding potential...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50554887(CHEMBL4778777)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516339(CHEMBL4461702)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516309(CHEMBL4594009)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516311(CHEMBL4516107)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50516335(CHEMBL4476528)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587086(CHEMBL5076977)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at rat alpha3beta2 nAChR expressed in xenopus oocytes assessed as inhibition of Ach- induced response at -70 mV holding potential...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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