Affinity DataEC50: 0.700nMAssay Description:Inverse agonist activity at GABAA alpha5beta3gamma2 in Homo sapiens (human) L(tk-) cells by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Effective concentration against human Alpha5-beta3-gamma2 GABA-A receptor was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Binding affinity to human alpha5beta3gamma2 GABA receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Binding affinity to human alpha5beta3gamma2 GABA receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 206nMAssay Description:Binding affinity to human alpha5beta3gamma2 GABA receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 455nMAssay Description:Binding affinity to human alpha5beta3gamma2 GABA receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.13E+3nMAssay Description:Binding affinity to human alpha5beta3gamma2 GABA receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Effective agonist dose for human Gamma-aminobutyric-acid A receptor alpha4-beta3-gamma2More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity on human Gamma-aminobutyric-acid A receptor alpha3-beta3-gamma2 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: >2.40E+4nMAssay Description:Displacement of [3H]-flumazenil from human GABA-A receptor alpha5beta3gamma2 expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+4nMAssay Description:Effective agonist dose for human Gamma-aminobutyric-acid A receptor alpha6-beta3-gamma2More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+5nMAssay Description:Effective agonist dose for human Gamma-aminobutyric-acid A receptor alpha5-beta3-gamma2 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+5nMAssay Description:Antagonistic potency against human Gamma-aminobutyric-acid A receptor alpha3-beta3-gamma2 expressed in Xenopus oocytes at 1 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+5nMAssay Description:Effective agonist dose for human Gamma-aminobutyric-acid A receptor alpha1-beta3-gamma2 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90E+5nMAssay Description:Agonist activity on human Gamma-aminobutyric-acid A receptor alpha3-beta3-gamma2 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+6nMAssay Description:Effective agonist dose for human Gamma-aminobutyric-acid A receptor alpha5-beta3-gamma2 expressed in Xenopus oocytesMore data for this Ligand-Target Pair