Compile Data Set for Download or QSAR
Report error Found 137 of ic50 for UniProtKB: P04757
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567433BDBM50567433(CHEMBL4869892)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238606BDBM50238606(CHEMBL4099865)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current at -70 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445330BDBM50445330(CHEMBL3104243)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567430BDBM50567430(CHEMBL4860756)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567432BDBM50567432(CHEMBL4876825)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567431BDBM50567431(CHEMBL4878931)
Affinity DataIC50: 3nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459664BDBM50459664(CHEMBL4218406)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459654BDBM50459654(CHEMBL4206157)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516340BDBM50516340(CHEMBL4439678)
Affinity DataIC50: 13nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567426BDBM50567426(CHEMBL4878856)
Affinity DataIC50: 15nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516316BDBM50516316(CHEMBL4454928)
Affinity DataIC50: 18nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459656BDBM50459656(CHEMBL4214931)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567413BDBM50567413(CHEMBL4865365)
Affinity DataIC50: 21nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459653BDBM50459653(CHEMBL4211045)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459661BDBM50459661(CHEMBL4215453)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238616BDBM50238616(CHEMBL3104238)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86240BDBM86240(Gly-L-Cys(1)-L-Cys(2)-L-Ser-L-Asn-L-Pro-L-Val-L-Cy...)
Affinity DataIC50: 32nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445331BDBM50445331(CHEMBL3104245)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238610BDBM50238610(CHEMBL4062759)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238580BDBM50238580(CHEMBL4099451)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238589BDBM50238589(CHEMBL4061135)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238579BDBM50238579(CHEMBL4070842)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567438BDBM50567438(CHEMBL4865866)
Affinity DataIC50: 44nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567427BDBM50567427(CHEMBL4872474)
Affinity DataIC50: 45nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238607BDBM50238607(CHEMBL4069809)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238611BDBM50238611(CHEMBL4097007)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459660BDBM50459660(CHEMBL4206670)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567405BDBM50567405(CHEMBL4867074)
Affinity DataIC50: 57nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238582BDBM50238582(CHEMBL4105157)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567437BDBM50567437(CHEMBL4871260)
Affinity DataIC50: 58nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516333BDBM50516333(CHEMBL4474223)
Affinity DataIC50: 60nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238585BDBM50238585(CHEMBL4071400)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516313BDBM50516313(CHEMBL4459917)
Affinity DataIC50: 64nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567414BDBM50567414(CHEMBL4851682)
Affinity DataIC50: 65nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238581BDBM50238581(CHEMBL4081435)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516315BDBM50516315(CHEMBL4515208)
Affinity DataIC50: 87nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445331BDBM50445331(CHEMBL3104245)
Affinity DataIC50: 94nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-induced current after 2 to 4 days by vol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516314BDBM50516314(CHEMBL4462168)
Affinity DataIC50: 95nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238617BDBM50238617(CHEMBL4091711)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516342BDBM50516342(CHEMBL4461998)
Affinity DataIC50: 113nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567411BDBM50567411(CHEMBL4856451)
Affinity DataIC50: 119nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445326BDBM50445326(CHEMBL3104239)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516306BDBM50516306(CHEMBL4438403)
Affinity DataIC50: 137nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238609BDBM50238609(CHEMBL4100403)
Affinity DataIC50: 147nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current at -80 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445326BDBM50445326(CHEMBL3104239)
Affinity DataIC50: 148nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567409BDBM50567409(CHEMBL4867777)
Affinity DataIC50: 175nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459659BDBM50459659(CHEMBL4214003)
Affinity DataIC50: 178nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238584BDBM50238584(CHEMBL4089797)
Affinity DataIC50: 178nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516327BDBM50516327(CHEMBL4538537)
Affinity DataIC50: 180nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567410BDBM50567410(CHEMBL4847671)
Affinity DataIC50: 191nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
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