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Found 3 of ic50 for UniProtKB: P42336
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/delta isoform(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM36408(1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1H-pyrazolo[3...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/delta isoform(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM36411(2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/delta isoform(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM618551(US11759530, Compound Table1.10)
Affinity DataIC50:  2.00E+7nMAssay Description:No assay is defined.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent