Compile Data Set for Download or QSAR
Report error Found 15 of ki for UniProtKB: P21918
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  5.10nMAssay Description:In vitro inhibition of [3H]-Spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranes (using L-tartrate salt of authentic rac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  8.70nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228777(CHEMBL80127)
Affinity DataKi:  17nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228772(CHEMBL418922)
Affinity DataKi:  41nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228774(CHEMBL80126)
Affinity DataKi:  89nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50134526(2-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl...)
Affinity DataKi:  120nMAssay Description:Ability to inhibit the binding of human DP receptor to PGD-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228776(CHEMBL81778)
Affinity DataKi:  130nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228771(CHEMBL312602)
Affinity DataKi:  159nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50159788(CHEMBL3786973)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to dopamine receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50187377(N-(3-(4-(4-(cyclohexylmethylsulfonamido)butyl)pipe...)
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity to dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228775(CHEMBL77448)
Affinity DataKi:  2.61E+3nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50228773(CHEMBL2021339)
Affinity DataKi:  2.62E+3nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Dopamine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50132104(6-Methoxy-1-methyl-4,9-dihydro-3H-beta-carboline |...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Dopamine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50136493(1-methyl-4,9-dihydro-3H-pyrido[3,4-b]indole | 1-Me...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Dopamine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed