Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ec50 for monomerid = 21138
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21138((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  0.220nM ΔG°:  -55.1kJ/mole EC50:  5.90nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21138((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  150nM EC50:  8nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona Tucson

LigandPNGBDBM21138((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  7.80nM ΔG°:  -46.3kJ/mole EC50:  12nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed