Affinity DataEC50: 12nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 355nMAssay Description:Inverse agonist activity at RORgamma in C57BL/6 mouse splenocytes assessed as reduction of IL-17 production after 2 days by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Inverse agonist activity at RORalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PXR (unknown origin)More data for this Ligand-Target Pair