TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 359nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 806nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair