Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ec50 for monomerid = 50194147
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50194147(4-Thio-UDP | CHEMBL384992 | [(2R,3S,4R,5R)-3,4-dih...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50194147(4-Thio-UDP | CHEMBL384992 | [(2R,3S,4R,5R)-3,4-dih...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50194147(4-Thio-UDP | CHEMBL384992 | [(2R,3S,4R,5R)-3,4-dih...)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating Gq protein assessed as [3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed