Affinity DataEC50: 6.5nMAssay Description:Agonist activity at human MOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
Affinity DataEC50: 6.70nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
Affinity DataEC50: 177nMAssay Description:Agonist activity at human DOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
Affinity DataEC50: 359nMAssay Description:Agonist activity at human MOR expressed in human U2OS cells assessed as increase in beta arrestin2 recruitment incubated for 90 mins by pathhunter be...More data for this Ligand-Target Pair
Affinity DataEC50: 424nMAssay Description:Agonist activity at human KOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair