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Found 5 of ic50 for monomerid = 27721
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
Fujisawa Pharmaceutical

LigandPNGBDBM27721(3-(4-cyanophenyl)quinoxaline-5-carboxamide | CHEMB...)
Affinity DataIC50:  8nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute

Curated by ChEMBL
LigandPNGBDBM27721(3-(4-cyanophenyl)quinoxaline-5-carboxamide | CHEMB...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PARP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute

Curated by ChEMBL
LigandPNGBDBM27721(3-(4-cyanophenyl)quinoxaline-5-carboxamide | CHEMB...)
Affinity DataIC50:  101nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute

Curated by ChEMBL
LigandPNGBDBM27721(3-(4-cyanophenyl)quinoxaline-5-carboxamide | CHEMB...)
Affinity DataIC50:  101nMpH: 8.0 T: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute

Curated by ChEMBL
LigandPNGBDBM27721(3-(4-cyanophenyl)quinoxaline-5-carboxamide | CHEMB...)
Affinity DataIC50:  101nMAssay Description:Inhibition of human recombinant PARP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed