Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 35604
LigandPNGBDBM35604(pyrazolo pyrimidine, 5j)
Affinity DataIC50:  2.77E+3nMT: 2°CAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM35604(pyrazolo pyrimidine, 5j)
Affinity DataIC50:  7.30E+3nMpH: 7.4 T: 2°CAssay Description:The enzyme was assayed in DELFIA format using purified FLAG-TOR in kinase buffer containing ATP and His6-S6K in the presence of inhibitor compounds. ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed