Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 373040
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Peloton Therapeutics

Curated by ChEMBL
LigandPNGBDBM373040(US10597366, Compound 289 | US9896418, Compound 289)
Affinity DataIC50:  9nMAssay Description:Inhibition of N-(3-Chlorophenyl-4,6-t2)-4-nitrobenzo[c][1,2,5]oxadiazol-5-amine binding to his-tagged HIF-2alpha PAS-B domain (unknown origin) measur...More data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Peloton Therapeutics

Curated by ChEMBL
LigandPNGBDBM373040(US10597366, Compound 289 | US9896418, Compound 289)
Affinity DataIC50:  10nMAssay Description:HIF-2a: The total assay volume was about 100 uL in the following configuration: 2 uL compound in 100% DMSO, 88 uL buffer with protein and probe and 1...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peloton Therapeutics

Curated by ChEMBL
LigandPNGBDBM373040(US10597366, Compound 289 | US9896418, Compound 289)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human ERG expressed in mammalian expression system by Q-patch clamp electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed