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Found 3 of ic50 for monomerid = 426342
LigandPNGBDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataIC50: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter. In general titrations were performed by titrating the protein (50 μM) to the te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataIC50: <300nMAssay Description:The biochemical activity assay for PDHK2 is based on the inactivation of PDC through phosphorylation by PDHK2. The assay is run in two steps: the enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataIC50: <300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent